Saiah, M. K. Eddine: search on Z-Library

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1

Chemistry and Pharmacology of the Piperidine-Based Analogues of Cocaine. Identification of Potent DAT Inhibitors Lacking the Tropane Skeleton

Kozikowski, Alan P., Araldi, Gian Luca, Boja, John, Meil, William M., Johnson, Kenneth M., Flippen-Anderson, Judith L., George, Clifford, Saiah, Eddine

Journal:

Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 232 KB

english, 1998

2

Small Molecules That Target Protein Misfolding

Gavrin, Lori Krim, Denny, Rajiah Aldrin, Saiah, Eddine

Journal:

Journal of Medicinal Chemistry

Year:

2012

Language:

english

File:

PDF, 3.01 MB

english, 2012

3

Direct Trifluoromethylation of Nitriles Promoted by Tetrabutylammonium Bifluoride

Huang, Adrian, Li, Huan-Qiu, Massefski, Walter, Saiah, Eddine

Journal:

Year:

2009

Language:

english

File:

PDF, 87 KB

english, 2009

4

Coupling structure-based design with combinatorial chemistry: application of active site derived pharmacophores with informative library design

John E. Eksterowicz, Erik Evensen, Christian Lemmen, G. Patrick Brady, J. Kevin Lanctot, Erin K. Bradley, Eddine Saiah, Leslie A. Robinson, Peter D.J. Grootenhuis, Jeffrey M. Blaney

Journal:

Journal of Molecular Graphics and Modelling

Year:

2002

Language:

english

File:

PDF, 345 KB

english, 2002

5

Discovery of NV-5138, the first selective Brain mTORC1 activator

Sengupta, Shomit, Giaime, Emilie, Narayan, Sridhar, Hahm, Seung, Howell, Jessica, O’Neill, David, Vlasuk, George P., Saiah, Eddine

Journal:

Scientific Reports

Year:

2019

File:

PDF, 3.27 MB

2019

6

N-Arylation of a hindered indoline as a route to 2-(2-methyl-1-(4-oxo-3,4-dihydrophthalazin-1-yl)-1H-indol-3-yl)acetic acid derivatives

Nikolaos Papaioannou, Vasilios Marathias, Zhao-Kui Wan, Neelu Kaila, Zahid Ali, Eddine Saiah

Journal:

Tetrahedron Letters

Year:

2011

Language:

english

File:

PDF, 549 KB

english, 2011

7

Approaches to discover non-ATP site kinase inhibitors

Gavrin, Lori Krim, Saiah, Eddine

Journal:

Year:

2013

Language:

english

File:

PDF, 467 KB

english, 2013

8

Phosphonium-mediated cyclization of N-(2-aminophenyl)thioureas: efficient synthesis of 2-aminobenzimidazoles

Zhao-Kui Wan, Erena Farah Ousman, Nikolaos Papaioannou, Eddine Saiah

Journal:

Tetrahedron Letters

Year:

2011

Language:

english

File:

PDF, 1.43 MB

english, 2011

9

Ketene Dithioacetals in the Aza-Diels−Alder Reaction with N -Arylimines: A Versatile Approach to Tetrahydroquinolines, 2,3-Dihydro-4-quinolones, and 4-Quinolones

Cheng, Dai, Zhou, Jinglan, Saiah, Eddine, Beaton, Graham

Journal:

Organic Letters

Year:

2002

Language:

english

File:

PDF, 80 KB

english, 2002

10

ChemInform Abstract: Phosphonium-Mediated Cyclization of N-(2-Aminophenyl)thioureas: Efficient Synthesis of 2-Aminobenzimidazoles.

Zhao-Kui Wan, Erena Farah Ousman, Nikolaos Papaioannou, Eddine Saiah

Journal:

Year:

2011

File:

PDF, 42 KB

2011

11

Informative Library Design as an Efficient Strategy to Identify and Optimize Leads: Application to Cyclin-Dependent Kinase 2 Antagonists

Bradley, Erin K., Miller, Jennifer L., Saiah, Eddine, Grootenhuis, Peter D. J.

Journal:

Journal of Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 77 KB

english, 2003

12

Rhodium-catalysed redox isomerization of hydroxy alkynes to trans keto and hydroxy vinyl esters. A short and stereoselective synthesis of dipeptide isosters

M.K. Eddine Saïah, Roberto Pellicciari

Journal:

Tetrahedron Letters

Year:

1995

Language:

english

File:

PDF, 209 KB

english, 1995

13

Chemistry and Biology of the 2.beta.-Alkyl-3.beta.-phenyl Analogs of Cocaine: Subnanomolar Affinity Ligands That Suggest a New Pharmacophore Model at the C-2 Position

Kozikowski, Alan P., Saiah, M. K. Eddine, Johnson, Kenneth M., Bergmann, John S.

Journal:

Journal of Medicinal Chemistry

Year:

1995

Language:

english

File:

PDF, 1.05 MB

english, 1995

14

Synthesis of Potent and Orally Efficacious 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitor HSD-016

Wan, Zhao-Kui, Chenail, Eva, Li, Huan-Qiu, Kendall, Christopher, Wang, Youchu,, Gingras, Stéphane, Xiang, Jason, Massefski, Walter W., Mansour, Tarek, S., Saiah, Eddine

Journal:

Journal of Organic Chemistry

Year:

2011

Language:

english

File:

PDF, 1.20 MB

english, 2011

15

Comparative Pharmacokinetics and Metabolism Studies in Lean and Diet- Induced Obese Mice: An Animal Efficacy Model for 11β -Hydroxysteroid Dehydrogenase Type 1 (11β -HSD1) Inhibitors

Wang, Mengmeng, Tian, Xianbin, Leung, Louis, Wang, Jianyao, Houvig, Nicole, Xiang, Jason, Saiah, Eddine, Hahm, Seung, Suri, Vipin, Xu, Xin

Journal:

Drug Metabolism Letters

Year:

2011

Language:

english

File:

PDF, 378 KB

english, 2011

16

Recent developments in targeting protein misfolding diseases

Denny, Rajiah Aldrin, Gavrin, Lori Krim, Saiah, Eddine

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2013

Language:

english

File:

PDF, 1.33 MB

english, 2013

17

ChemInform Abstract: Direct Trifluoromethylation of Nitriles Promoted by Tetrabutylammonium Bifluoride.

Adrian Huang, Huan-Qiu Li, Walter Massefski, Eddine Saiah

Journal:

Year:

2010

File:

PDF, 27 KB

2010

18

Discovery and gram-scale synthesis of BMS-593214, a potent, selective FVIIa inhibitor

Priestley, E. Scott, De Lucca, Indawati, Zhou, Jinglan, Zhou, Jiacheng, Saiah, Eddine, Stanton, Robert, Robinson, Leslie, Luettgen, Joseph M., Wei, Anzhi, Wen, Xiao, Knabb, Robert M., Wong, Pancras C.

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2013

Language:

english

File:

PDF, 542 KB

english, 2013

19

Small Molecule Coagulation Cascade Inhibitors in the Clinic

Saiah, Eddine, Soares, Chris

Journal:

Current Topics in Medicinal Chemistry

Year:

2005

Language:

english

File:

PDF, 148 KB

english, 2005

20

Structure-Activity Relationship Studies of N-Sulfonyl Analogs of Cocaine: Role of Ionic Interaction in Cocaine Binding

Kozikowski, Alan P., Saiah, M. K. Eddine, Bergmann, John S., Johnson, Kenneth M.

Journal:

Journal of Medicinal Chemistry

Year:

1994

Language:

english

File:

PDF, 433 KB

english, 1994

21

The Role of 11Beta-Hydroxysteroid Dehydrogenase in Metabolic Disease and Therapeutic Potential of 11Beta-HSD1 Inhibitors

Journal:

Current Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 297 KB

english, 2008

22

Ketene Dithioacetals in the Aza-Diels—Alder Reaction with N-Arylimines: A Versatile Approach to Tetrahydroquinolines, 2,3-Dihydro-4-quinolones, and 4-Quinolones.

Dai Cheng, Jinglan Zhou, Eddine Saiah, Graham Beaton

Journal:

Year:

2003

Language:

english

File:

PDF, 251 KB

english, 2003

23

A small molecule inhibitor of Rheb selectively targets mTORC1 signaling

Mahoney, Sarah J., Narayan, Sridhar, Molz, Lisa, Berstler, Lauren A., Kang, Seong A., Vlasuk, George P., Saiah, Eddine

Journal:

Nature Communications

Year:

2018

Language:

english

File:

PDF, 1.82 MB

english, 2018

24

Probing acid replacements of thiophene PTP1B inhibitors

Zhao-Kui Wan, Bruce Follows, Steve Kirincich, Douglas Wilson, Eva Binnun, Weixin Xu, Diane Joseph-McCarthy, Junjun Wu, Michael Smith, Yan-Ling Zhang, May Tam, David Erbe, Steve Tam, Eddine Saiah, Jinb

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2007

Language:

english

File:

PDF, 343 KB

english, 2007

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